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A kinetic view of GPCR allostery and biased agonism

Lane JR, May LT, Parton RG, Sexton PM, Christopoulos A. A kinetic view of GPCR allostery and biased agonism. Nat Chem Biol 13, 929–937, 2017. https://doi.org/10.1038/nchembio.2431