Discovery of a positive allosteric modulator of cholecystokinin action at CCK1R in normal and elevated cholesterol

Harikumar KG, Coudrat T, Desai AJ, Dong M, Dengler DG, Furness SGB, Christopoulos A, Wootten D, Sergienko EA, Sexton PM, Miller LJ. Discovery of a positive allosteric modulator of cholecystokinin action at CCK1R in normal and elevated cholesterol. Frontiers in Endocrinology 12:789957, 2021. https://doi.org/10.3389/fendo.2021.789957